
Rilmenidine Phosphate
CAS No. 85409-38-7
Rilmenidine Phosphate ( —— )
产品货号. M19181 CAS No. 85409-38-7
Rilmenidine Phosphate 是一种选择性 I(1) 咪唑啉受体激动剂,用于治疗高血压。
纯度: >98% (HPLC)






规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥648 | 有现货 |
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10MG | ¥1126 | 有现货 |
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25MG | ¥2252 | 有现货 |
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50MG | ¥3556 | 有现货 |
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100MG | ¥5338 | 有现货 |
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500MG | ¥11097 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Rilmenidine Phosphate
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Rilmenidine Phosphate 是一种选择性 I(1) 咪唑啉受体激动剂,用于治疗高血压。
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产品描述Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.(In Vitro):Rilmenidine provides antihypertensive efficacy comparable with that of diuretics, beta-blockers, calcium channel blockers, and angiotensin-converting enzyme (ACE) inhibitors.Rilmenidine phosphate (25-100 μM; 24 hours) inhibits K562 cell proliferation.(In Vivo):Rilmenidine phosphate-treated N171-82Q mice (i.p.; 4-times a week) displays significant improved forelimb grip strength and all limbs grip strength from 12 to 22 weeks of age.Rilmenidine phosphate decreases levels of mutant huntingtin.
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体外实验Rilmenidine provides antihypertensive efficacy comparable with that of diuretics, beta-blockers, calcium channel blockers, and angiotensin-converting enzyme (ACE) inhibitors.Rilmenidine phosphate (25-100 μM; 24 hours) inhibits K562 cell proliferation. Cell Proliferation Assay Cell Line:K562 cells Concentration:25, 50, 100 μM Incubation Time:24 hours Result:Dose-dependently inhibited K562 colony formation.
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体内实验Rilmenidine phosphate-treated N171-82Q mice (i.p.; 4-times a week) displays significant improved forelimb grip strength and all limbs grip strength from 12 to 22 weeks of age.Rilmenidine phosphate decreases levels of mutant huntingtin.
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同义词——
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通路Others
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靶点Other Targets
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受体I(1) imidazoline receptor
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研究领域Others-Field
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适应症——
化学信息
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CAS Number85409-38-7
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分子量278.24
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分子式C10H19N2O5P
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纯度>98% (HPLC)
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溶解度In Vitro:?H2O : 83.33 mg/mL (299.49 mM)
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SMILESC1CC1C(C1CC1)NC1=NCCO1.OP(=O)(O)O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Srdic-Rajic T, et al.Eur J Pharm Sci. 2016 Jan 1;81:172-80.
产品手册




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